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Irinotecan

Metastatic Malignant Neoplasm In The Brain

Explore 101 assets in Metastatic Malignant Neoplasm In The Brain
Floatz Rating
B63/100
Confidence
Indicative
v0.2
Sponsor
Tianjin Medical University Cancer Institute and Hospital
Modality
Small molecule
Development Phase
Phase 3
Status
Active
Evidence ledger · v0.2

Clinical Evidence

Clinical track record: trial progression, reported outcomes, safety signals, and endpoint quality.
58High confidence
Detailed axis rationale is planned and will be published soon.
TrialPhaseStatusNPrimary endpointReadout
A Phase II Clinical Study of Utidelone and Bevacizumab With or Without Etoposide in Patients With Brain Metastases From Malignant Solid Tumors
Not Yet Recruiting
Sac-TMT Combined With Bevacizumab in TNBC With Brain Metastases
Recruiting
Study of SHR-A1811 Combined With Pyrotinib and Bevacizumab in Advanced Breast Cancer With Brain Metastasis
Recruiting
Safety and Efficacy of NEO212 in Patients With Astrocytoma IDH-mutant, Glioblastoma IDH-wildtype or Brain Metastasis
Recruiting
Combination Liposomal Irinotecan and Pembrolizumab For Triple-Negative Breast Cancer (TNBC) With Brain Metastases (BM)
Withdrawn
Phase 1/2 Trial of S241656 in Selected RAS/MAPK Mutation- Positive Malignancies
Recruiting
Osimertinib With or Without Bevacizumab in Treating Patients With EGFR Positive Non-small Cell Lung Cancer and Brain Metastases
Active Not Recruiting
Bevacizumab and Atezolizumab With or Without Cobimetinib in Treating Patients With Untreated Melanoma Brain Metastases
Active Not Recruiting
A Study Evaluating INIPARIB in Combination With Chemotherapy to Treat Triple Negative Breast Cancer Brain Metastasis
Completed
Study of the Combination of Vorinostat and Radiation Therapy for the Treatment of Patients With Brain Metastases
Completed

Competitive Position

Competitive setting: how crowded the indication is, class-level failures, and timing against rivals.
73High confidence
Detailed axis rationale is planned and will be published soon.

Same indication · Metastatic Malignant Neoplasm In The Brain

AssetSponsorPhaseRating
Irinotecan (this asset)Tianjin Medical University Cancer Institute and HospitalP3B · 63
TrastuzumabIambic Therapeutics, IncP4BB
IcotinibBetta Pharmaceuticals Co., Ltd.P3BB
Trastuzumab DeruxtecanBaptist Health South FloridaP4BB
Copper Cu 64-Dota-TrastuzumabCity of Hope Medical CenterP4BB
CapecitabineCancer Institute and Hospital, Chinese Academy of Medical SciencesP3BB
MemantineNRG OncologyP3BB
RegorafenibNeonc Technologies, Inc.P2BB
GefitinibAlpha Biopharma (Jiangsu) Co., Ltd.P3B

+42 more in the Metastatic Malignant Neoplasm In The Brain cohort

Other indications for Irinotecan

IndicationSponsorPhaseRating
Rectal CancerP4BBB · 78
Exocrine Pancreatic CarcinomaP2/3BBB · 78
Colon AdenocarcinomaP3BBB · 76

Scientific Foundation

Strength of the underlying biology: target validation, tractability, modality fit, and how related mechanisms have fared.
NR

Planned for methodology v0.2.

Development Feasibility

How realistically the program can be executed, drawing on modality precedent, enrollment dynamics, and sponsor delivery.
NR

Planned for methodology v0.2.

Commercial Opportunity

Commercial prize: addressable population, unmet need, and the value case for the indication.
NR

Planned for methodology v0.2.

IP & Exclusivity

Exclusivity position, covering patent protection and freedom-to-operate runway.
NR

Planned for methodology v0.2.

Manufacturing & Supply

Manufacturing and supply readiness, driven by modality process and scale-up risk.
NR

Planned for methodology v0.2.

Related assets

Citation

Floatz Terminal. Irinotecan in Metastatic Malignant Neoplasm In The Brain. Methodology v0.2.
Rated under v0.2 effective July 8, 2026. Last refreshed July 8, 2026.
Accessed July 14, 2026.
https://terminal.floatz.ai/assets/irinotecan-metastatic-malignant-neoplasm-in-the-brain

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