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Neratinib

HER2 Positive Breast Carcinoma

Explore 176 assets in HER2 Positive Breast Carcinoma
Floatz Rating
B57/100
Confidence
Indicative
v0.2
Sponsor
Fudan University
Modality
Small molecule
Development Phase
Phase 3
Status
Active
Evidence ledger · v0.2

Clinical Evidence

Clinical track record: trial progression, reported outcomes, safety signals, and endpoint quality.
53High confidence
Detailed axis rationale is planned and will be published soon.
TrialPhaseStatusNPrimary endpointReadout
T-DXd With or Without Neratinib for HER2 Positive Breast Cancer With Brain Metastasis
Not Yet Recruiting
Neratinib in Extended Adjuvant Treatment for HER2+ Early Breast Cancer With pCR But High-Risk Features: A Hebei Multi-Center Real-World Study
Not Yet Recruiting
Adjuvant Trastuzumab Plus Neratinib in Hormone Receptor-Positive/Human Epidermal Growth Factor Receptor 2-Positive Breast Cancer After Neoadjuvant Trastuzumab Plus Pertuzumab
Recruiting
Kadcyla And Neratinib for Interception of HER2+ Breast Cancer With Molecular Residual Disease
Recruiting
Three Antidiarrheal Strategies in HER2+/HR+ Early Breast Cancer Patients Treated With Extended Adjuvant Neratinib
Active Not Recruiting
Trial of Pre-operative Neratinib and Endocrine Therapy With Trastuzumab in ER-Positive, HER-2 Positive Breast Cancers
Recruiting
Neratinib Dose Escalation Regimen for HER2 Positive Early Breast Cancer
Unknown
A Study to Characterize Colon Pathology in Patients With HER2 Amplified Breast Cancer Treated With Neratinib
Completed
Evaluating the Efficacy of Neratinib on Live Cell HER2 Signaling Transduction Analysis Positive Triple Negative Breast
Unknown
Adjuvant Therapy With Neratinib in HER2 Positive Early Breast Cancer
Recruiting
Show 5 more trials
Incidence and Severity of Diarrhea in Patients With HER2 Positive Breast Cancer Treated With Trastuzumab and Neratinib
Completed
Neratinib in Treating Older Patients With Stage IV HER2-Positive Breast Cancer
Completed
An Open-Label Study to Characterize the Incidence and Severity of Diarrhea in Patients With Early-Stage HER2+ Breast Cancer Treated With Neratinib and Loperamide
Completed
A Study of Neratinib Plus Capecitabine Versus Lapatinib Plus Capecitabine in Patients With HER2+ Metastatic Breast Cancer Who Have Received Two or More Prior HER2 Directed Regimens in the Metastatic Setting
Completed
I-SPY TRIAL: Neoadjuvant and Personalized Adaptive Novel Agents to Treat Breast Cancer
Recruiting

Competitive Position

Competitive setting: how crowded the indication is, class-level failures, and timing against rivals.
65High confidence
Detailed axis rationale is planned and will be published soon.

Same indication · HER2 Positive Breast Carcinoma

AssetSponsorPhaseRating
Neratinib (this asset)Fudan UniversityP3B · 57
TrastuzumabSWOG Cancer Research NetworkP4BB
PertuzumabSWOG Cancer Research NetworkP4BB
RibociclibDanish Breast Cancer Cooperative GroupP3BB
DocetaxelOhio State University Comprehensive Cancer CenterP3BB
CyclophosphamideNational University Hospital, SingaporeP3BB
CapecitabineMedSIRP4BB
Vinorelbine DitartrateFudan UniversityP3BB
gb221Genor Biopharma Co., Ltd.P3BB

+42 more in the HER2 Positive Breast Carcinoma cohort

Other indications for Neratinib

IndicationSponsorPhaseRating
Breast CarcinomaP2BB · 65
Breast CancerP3B · 60
Breast NeoplasmP3B · 60

Scientific Foundation

Strength of the underlying biology: target validation, tractability, modality fit, and how related mechanisms have fared.
NR

Planned for methodology v0.2.

Development Feasibility

How realistically the program can be executed, drawing on modality precedent, enrollment dynamics, and sponsor delivery.
NR

Planned for methodology v0.2.

Commercial Opportunity

Commercial prize: addressable population, unmet need, and the value case for the indication.
NR

Planned for methodology v0.2.

IP & Exclusivity

Exclusivity position, covering patent protection and freedom-to-operate runway.
NR

Planned for methodology v0.2.

Manufacturing & Supply

Manufacturing and supply readiness, driven by modality process and scale-up risk.
NR

Planned for methodology v0.2.

Related assets

Citation

Floatz Terminal. Neratinib in HER2 Positive Breast Carcinoma. Methodology v0.2.
Rated under v0.2 effective July 8, 2026. Last refreshed July 8, 2026.
Accessed July 14, 2026.
https://terminal.floatz.ai/assets/neratinib-her2-positive-breast-carcinoma

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